Pregnenolone

Pregnenolone is a neurosteroid and steroid hormone precursor, synthesized from cholesterol. It’s the first step in the steroid hormone cascade.

🧠 Key Physiological Functions of Pregnenolone

1. Hormone Precursor

  • Acts as a building block for:
    • Progesterone
    • Cortisol
    • Aldosterone
    • Testosterone
    • Estrogens
    • DHEA
  • Essential for maintaining hormonal balance in the body.

2. Brain & Nervous System Effects

  • Neurosteroid activity: Synthesized in the brain, it modulates:
    • Synaptic transmission
    • Neuroplasticity
    • Myelination
  • Influences mood, motivation, and cognitive function.

3. Memory & Cognitive Enhancement

  • Animal and limited human studies suggest it may:
    • Enhance memory formation
    • Improve learning capacity
    • Protect against neurodegeneration
  • Protects brain cells from injury and oxidative stress.
  • Thought to modulate NMDA and GABA-A receptors, affecting excitability and inhibition in the brain.

4. Anti-fatigue & Stress Modulation

  • May help the body cope with stress by supporting adrenal hormone production (e.g., cortisol).
  • Possibly improves energy levels and resilience under stress.
  • May have anti-anxiety and antidepressant effects by modulating brain neurotransmitters.

5. Immune System Modulation

  • Some evidence suggests pregnenolone may influence immune responses, although this is less understood.

🧬 Where Is It Made?

  • Adrenal glands, gonads, brain, liver, and retina.

⚖️ Clinical Relevance

  • Levels decline with age.
  • Studied (but not definitively proven) for potential roles in:
    • Alzheimer’s disease
    • Depression
    • Schizophrenia
    • Fatigue syndromes
    • Hormonal deficiencies

📉 Decline With Age

  • Pregnenolone levels peak in early adulthood and decline significantly with age, potentially affecting hormone balance, memory, and energy.